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612-822-4611
Functional Selectivity of G Protein-Coupled Receptor Ligands: New Opportunities for Drug Discovery

Functional Selectivity of G Protein-Coupled Receptor Ligands: New Opportunities for Drug Discovery

Paperback

Series: Receptors

Medical ReferenceAnatomy & Physiology

ISBN10: 1493961160
ISBN13: 9781493961160
Publisher: Humana Pr
Published: Aug 23 2016
Pages: 292
Weight: 0.94
Height: 0.64 Width: 6.14 Depth: 9.21
Language: English
Historical Overview of the Concept of Functional Selectivity.- Functional Selectivity: Theoretical Considerations and Future Directions.- Agonist Selective Coupling of G Protein-Coupled Receptors.- Ligand-Selective Receptor Desensitization and Endocytosis.- Selectivity for G protein or Arrestin-Mediated Signaling.- In Vivo Evidence for and Consequences of Functional Selectivity.- Functional Selectivity at Adrenergic Receptors.- Signaling Diversity Mediated by Muscarinic Acetylcholine Receptor Subtypes and Evidence for Functional Selectivity.- Functional Selectivity at Serotonin Receptors.- Functional Selectivity at Dopamine Receptors.- Functional Selectivity at Receptors for Cannabinoids and other Lipids.- Functional Selectivity at Opioid Receptors Graciela Piñeyro.- Functional Selectivity at non-Opioid Peptide Receptors

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Anatomy & Physiology