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612-822-4611
P2y1-Retseptory

P2y1-Retseptory

Paperback

Medical Reference

Currently unavailable to order

ISBN10: 3659425613
ISBN13: 9783659425615
Publisher: Lap Lambert Academic Pub
Published: Jul 25 2013
Pages: 164
Weight: 0.55
Height: 0.38 Width: 6.00 Depth: 9.00
Language: Russian
Kniga posvyashchena voprosam sovremennogo pred-stavleniya o P2Y1-retseptorakh s opisaniem ikh znacheniya v sisteme gomeostaza, molekulyarnoy struktury P2Y1-retseptora, roli otdel'nykh ego sub-struktur v funktsional'noy aktivnosti, mekhanizma vzaimodeystviya ligandov s aktivnym tsentrom retseptora. Opisany fiziologicheskaya rol' dannogo retseptora i naibolee izuchennye k nastoyashchemu vremeni ego antagonisty. Podrobno izlozheny khimicheskiy sintez i svoystva novykh soedineniy klassov kondensirovannykh benzimidazolov i proizvodnykh aminospirtov ryada indola. Privodyatsya eksperimental'nye dannye dlya naibolee aktivnykh veshchestv s P2Y-antagonisticheskimi svoystvami ikh vliyanii na sosudisto-trombotsitarnyy i koagulyatsionnyy gemostaz, opisyvayutsya ikh antitromboticheskie svoystva. Rassmotreny komp'yuternye metody poiska novykh soedineniy s P2Y1-antagonisticheskoy aktivnost'yu.

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